高等学校化学学报

高等学校化学学报 ›› 2000, Vol. 21 ›› Issue (12): 1855.

• 研究简报 • 上一篇    下一篇

生物合理设计光系统Ⅱ抑制剂研究(Ⅵ)--2-氰基-3-甲硫基-3-烷氨(苄氨)基丙烯酸乙酯的合成及其Hill反应抑制活性

刘华银, 谭惠芬, 杨华铮   

  1. 南开大学元素, 有机化学研究所元素有机化学国家重点实验室, 天津 300071
  • 收稿日期:1999-12-04 出版日期:2000-12-24 发布日期:2000-12-24
  • 通讯作者: 杨华铮(1936年出生),女,教授,博士生导师,从事有机化学和农药化学研究.E-mail:yanghz@public.tpt.tj.cn E-mail:yanghz@public.tpt.tj.cn
  • 基金资助:

    国家自然科学基金(批准号:29832050;29702006);高等学校博士学科点专项科研基金资助

Studies on Bio-rational Molecular Design of Photosystem II Inhibitors——(Ⅵ) Synthesis and Hill Inhibitory Activity of Ethyl2-Cyano-3-methylthio-alkyl(benzyl)acrylates

LIU Hua-Yin, TAN Hui-Fen, YANG Hua-Zheng    

  1. State Key Laboratory and Institute of Elemento Organic Chemistry, Nankai University, Tianjin 300071, China
  • Received:1999-12-04 Online:2000-12-24 Published:2000-12-24

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关键词: D1蛋白, 丙烯酸乙酯, 合成, Hill反应抑制活性

Abstract: Based on targets structure and bio rational molecular design, the title compounds have been synthesized, all compounds have been confirmed by1H NMRand elemental analysis.The Hill reaction inhibitory activity of all the title compounds was tested and the bioassay results indicate that some of them show a good inhibitory activity, the relationship between the structure and inhibitory was analyzed

Key words: D1 protein, Ethyl acrylates, Synthesis, Hill inhibitory activity

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