高等学校化学学报 ›› 1995, Vol. 16 ›› Issue (2): 234.

• 研究简报 • 上一篇    下一篇

新型含噻二唑环磺酰脲的合成及其生物活性的研究

杨新玲, 陈馥衡   

  1. 北京农业大学应用化学系, 北京 100094
  • 收稿日期:1994-02-21 修回日期:1994-08-03 出版日期:1995-02-24 发布日期:1995-02-24
  • 通讯作者: 陈馥衡
  • 作者简介:杨新玲,女,27岁,博士研究生.

Synthesis of Some Novel Sulfonylureas Containing Thiadiazole and Their Biological Activity

YANG Xin-Ling, CHEN Fu-Heng   

  1. Department of Applied Chemistry, Beijing Agricultural Univiversity, Beijing, 100094
  • Received:1994-02-21 Revised:1994-08-03 Online:1995-02-24 Published:1995-02-24

关键词: 噻二唑, 磺酰脲, 合成, 生物活性

Abstract: Twenty-five novel sulfonylureas containing thiadiazole have been synthesized by treating 2-amino-5-subthiadiazole with sulfonylisocynate.Tlieir structures were confirmed by IR,1HNMR and elementary analysis.The preliminary biological test shows that compounds 1,2,5 and 22 are effective against broadleaf plants at 2.25 kg/ha in pre-or post-emergence;10,22,25 also exhibit certain fungicidal activity against puccinia Recondita at 0.125%in vivo.

Key words: Thiadiazole, Sulfonylurea, Synthesis, Biological activity

TrendMD: