高等学校化学学报

高等学校化学学报 ›› 2001, Vol. 22 ›› Issue (S1): 92.

• 研究论文 • 上一篇    下一篇

1-(2,4-二氯苯基)-1-氨基-4,4-二甲基-2-(1,2,4-三唑-1-基)-3-戊酮(醇)的合成及生物活性研究

刘建兵, 赵国锋, 李焜昶, 金桂玉   

  1. 南开大学元素有机化学研究所, 元素有机化学国家重点实验室, 天津 300071
  • 收稿日期:2001-07-17 出版日期:2001-12-31 发布日期:2001-12-31
  • 通讯作者: 金桂玉(1935年出生),女,教授,主要从事有机合成和农药化学研究.Tel:022-23509956.
  • 基金资助:

    国家自然科学基金(批准号:29832050)及"九五"攻关课题资助.

Studies on Syntheses and Biological Activities of 1H-1,2,4-Triazolo-1-yl Amine Compounds

LIU Jian-Bing, ZHAO Guo-Feng, LI Yu-Chang, JIN Gui-Yu   

  1. The State Key Ldboratory of Elemento-Organic Chemistry, Institute of Elemento-Organic Chemistry, Nankai University, Tianjin 300071, China
  • Received:2001-07-17 Online:2001-12-31 Published:2001-12-31

PDF (PC)

被引次数

1

摘要：

通过不同的胺对烯唑醇前体1的1,4-亲核加成反应,合成了目标化合物2,并将其还原得到了其还原产物3.生物活性测试结果发现,化合物3表现出较好的杀菌活性及一定程度的椬物生长调节活性.

关键词: 三唑, 1, 4-亲核加成反应, 生物活性

Abstract:

The title compounds 2 were prepared by 1, 4-nuclophilic addition different amine compounds to the precursor of diniconazole 1, which were reduced to give the compounds 3. From the screening results of biological activities, the compounds 3 possess good fungicidal and plant growth regulation activities to some degree, but low herbicidal activities.

Key words: Triazole, 1,4-Nuclophilic Addition, Biological Activities

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