Synthesis and Insecticidal Activities of New Pyrethroids Containing γ-Aryl Allyl Alcohol Moieties

Abstract

Abstract: Aseries of new pyrethroids containing γ-aryl allyl alcohol moieties were synthesized by using the esterification of 2,2-dimethyl-3-(2,2-dimethy vinyl)cyclopropane carbonyl chloride and 3-(2,2-dichlorovinyl)-2,2-dimethylcyclopropane carbonyl chloride with γ-aryl allyl alcohols. Their structures were confirmed by means of IR,¹HNMR,MS and elementary analysis.The preliminary biological test shows that some of the compounds have highly insecticidal activities,but the knock down activities against mosquito are lower than PY116.

Key words: γ-Aryl allyl alcohol, Pyrethroid, Insecticidal activity

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CHEN Ya-Juan, HUANG Run-Qij, MA Jun-An . Synthesis and Insecticidal Activities of New Pyrethroids Containing γ-Aryl Allyl Alcohol Moieties[J]. Chem. J. Chinese Universities, 1995, 16(4): 585.

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Synthesis and Insecticidal Activities of New Pyrethroids Containing γ-Aryl Allyl Alcohol Moieties

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