Synthesis and Bioactivity of 3-N-Benzyloxycarbonyl-β-aminobutyric Saccharide Carboxylate

Chem. J. Chinese Universities

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Synthesis and Bioactivity of 3-N-Benzyloxycarbonyl-β-aminobutyric Saccharide Carboxylate

ZANG Hong-Jun¹, LI Zheng-Ming²*, FAN Zhi-Jin², LIU Xiu-Feng², WANG Su-Hua²

1. Tianjin Municipal Key Laboratory of Fiber Modification & Functional Fiber, School of Material Science and Chemistry Engineering, Tianjin Polytechnic University, Tianjin 300160, China;
2. Key Labortary of Elemento-organic Chemisty, Institute of Elemento-organic Chemistry, Nankai University, Tianjin 300071, China

Received:2006-08-14 Revised:1900-01-01 Online:2007-08-10 Published:2007-08-10
Contact: LI Zheng-Ming

Abstract

Abstract: The plant activators such as D,L-β-aminobutyric acids can induce systemically acquired resiatance in the treated plants against the pathogen infection. Saccharide carboxylate compounds are known for their physiological and pharmaceutical importance. In order to investigate the synergic effect of the glucose and β-aminobutyric acid , eight new glycosyl esters of β-aminobutyric acid were synthesized with the reaction of 3-N-benzyloxycarbonyl-β-aminobutyric acid with acetylated glycosyl bromide or di-O-isopropyllidene-glucose. The structures were confirmed via elemental analysis and ¹H NMR. Bioassay results indicate that several compounds show a better induced activity against pathogen infection than salicylic acid.

Key words: D,L-β-Aminobutyric acid, Glucosyl ester, Induced resistance, Bioactivity

CLC Number:

O625

TrendMD:

ZANG Hong-Jun¹, LI Zheng-Ming²*, FAN Zhi-Jin², LIU Xiu-Feng², WANG Su-Hua². Synthesis and Bioactivity of 3-N-Benzyloxycarbonyl-β-aminobutyric Saccharide Carboxylate[J]. Chem. J. Chinese Universities, doi: .

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Synthesis and Bioactivity of 3-N-Benzyloxycarbonyl-β-aminobutyric Saccharide Carboxylate

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