Studies on the Synthesis of Phosphonodipeptides and Their Herbicidal Activity (Ⅱ)

Abstract

Abstract: It was reported in literature that phosphonodipeptides had significant biological activities.In order to look for new herbicides, a series of novel phosphonodipeptides have been prepared by the reaction of (PhO)₂P(O)CH₂NH₂ or (EtO)₂P(O)CH₂NH₂ with ClCH₂CONHCHR COOR'and ClCH₂CONHCHRP(O)(OPh)₂ separately in the presence of triethylamine in benzene.The structures of all the compounds prepared were proved by ¹H NMR, IR and MS.Their spectroscopic spectra and biological activities were discussed.It was found that some of them showed good herbicidal activity.

Key words: a-aminoalkyl phosphonate ester, Phosphonodipeptide, Herbicidal activity

TrendMD:

CHEN Ru-yu, ZHANG Yue-hua, CHENG Mu-ru . Studies on the Synthesis of Phosphonodipeptides and Their Herbicidal Activity (Ⅱ)[J]. Chem. J. Chinese Universities, 1992, 13(5): 611.

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Studies on the Synthesis of Phosphonodipeptides and Their Herbicidal Activity (Ⅱ)

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